Retatrutide 10mg98.5% Pure
GLP-1 Agonists

Retatrutide 10mg

A novel triple-agonist peptide targeting GLP-1, GIP, and glucagon receptors simultaneously, Retatrutide represents the cutting edge of incretin-based metabolic research compounds.

Molecular Weight

4979.57 g/mol

Sequence

Complex 39-amino acid sequence modified with fatty acid

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Molecular Formula

C221H347N61O66

Molecular Weight

4979.57 g/mol

Purity

98.5%

CAS Number

2381089-83-2

Half Life

6-7 days

Storage

2-8°C

Administration

subcutaneous

Research Status

phase2

View on PubChem

Description

Retatrutide is an innovative single-molecule triple agonist that activates three key metabolic receptors: glucagon-like peptide-1 (GLP-1), glucose-dependent insulinotropic polypeptide (GIP), and glucagon receptors. This multi-receptor approach represents an evolution in metabolic research tools, allowing scientists to investigate synergistic receptor activation patterns. Research literature has documented Retatrutide's unique pharmacological profile. Studies suggest the compound's triple-agonist mechanism may influence multiple metabolic pathways simultaneously—including glucose homeostasis, lipid metabolism, appetite signaling, and energy expenditure. Research Applications Triple receptor agonism studies Incretin pathway research Metabolic syndrome investigations Glucose homeostasis studies Energy expenditure research For qualified researchers conducting legitimate scientific investigations only.

Research

Retatrutide (Triple agonist) research: - Obesity treatment - Type 2 diabetes management - NASH (fatty liver disease) - Cardiovascular risk reduction - Metabolic syndrome - Appetite regulation - Energy expenditure - Lipid metabolism

Mechanism

Triple receptor agonist targeting: 1. GLP-1 receptor activation 2. GIP receptor activation 3. Glucagon receptor activation 4. Enhanced insulin secretion 5. Delayed gastric emptying 6. Increased energy expenditure 7. Improved lipid metabolism

Benefits

Significant weight loss (up to 24%) Improved glycemic control Reduced liver fat Better lipid profiles Cardiovascular benefits Appetite suppression Increased energy expenditure Metabolic flexibility

Dosage

Research dosing (Phase 2 trials): - Starting: 1mg weekly - Titration: Increase by 1mg every 4 weeks - Maintenance: 4-12mg weekly - Maximum: 12mg weekly - Duration: 48+ weeks in trials

Safety

Common side effects: - Nausea (dose-dependent) - Vomiting - Diarrhea - Constipation - Injection site reactions - Fatigue - Dizziness - Increased heart rate
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